SCHEMBL4767876

SCHEMBL4767876

NS(=O)(=O)CCc1cccc(Cl)c1Cl

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 2/20 0.58
PNMT P11086 1/20 0.53
IDO1 P14902 2/20 0.47
PTGES2 Q9H7Z7 2/20 0.43
AKR1B1 P15121 1/20 0.40
RECQL P46063 2/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 1/20 0.38
CD38 P28907 1/20 0.37
CA1 P00915 1/20 0.37
ACHE P22303 1/20 0.37
PTPRC P08575 1/20 0.37
PTPRG P23470 1/20 0.37
CYP2A13 Q16696 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6011891 0.81 TAAR1 (0.53) TAAR1PNMTIDO1PTGES2AKR1B1
SCHEMBL9390698 0.81 PNMT (0.57) TAAR1PNMTIDO1PTGES2AKR1B1
SCHEMBL10690855 0.74 TAAR1 (0.63) TAAR1PNMTIDO1RECQLKDM4E
SCHEMBL1570973 0.74 TAAR1 (1.00) TAAR1PNMTIDO1
SCHEMBL30785390 0.74 TAAR1 (1.00) TAAR1PNMTIDO1
SCHEMBL1462274 0.74 TAAR1 (0.37) TAAR1PNMTPTGES2RECQLALDH1A1
SCHEMBL25435653 0.71 TAAR1 (0.57) TAAR1IDO1AKR1B1RECQLTSHR
SCHEMBL27737597 0.71 RECQL (0.42) TAAR1PNMTPTGES2RECQLCA1
SCHEMBL2907991 0.71 PNMT (0.54) TAAR1PNMTIDO1AKR1B1KDM4E
SCHEMBL10914706 0.71 TAAR1 (0.77) TAAR1PNMTIDO1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP claimed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO claimed
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed