SCHEMBL4768412

SCHEMBL4768412

O=C(Nc1ccc2c(c1)CCN(C1CCC1)CC2)c1ccc2[nH]ccc2c1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.53
MAOB P27338 1/20 0.53
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
MAPT P10636 1/20 0.48
HRH3 Q9Y5N1 1/20 0.47
CHRNA7 P36544 1/20 0.46
PLAU P00749 1/20 0.46
EPHX1 P07099 1/20 0.44
ROCK2 O75116 1/20 0.44
ESR1 P03372 2/20 0.44
CHRM2 P08172 1/20 0.44
PRMT5 O14744 1/20 0.44
WDR77 Q9BQA1 1/20 0.44
HSD11B1 P28845 1/20 0.43
MELK Q14680 1/20 0.43
TMPRSS2 O15393 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4768268 0.94 SLC2A1 (0.47) MAOAMAOBNPC1RAB9AMAPT
SCHEMBL4768483 0.93 ALDH1A1 (0.51) MAOAMAOBNPC1RAB9AMAPT
Trifluoroacetic Acid SCHEMBL4772660 0.87 ESR1 (0.50) NPC1RAB9AMAPTHRH3CHRNA7
SCHEMBL4774628 0.83 TMPRSS2 (0.61) NPC1RAB9AMAPTHRH3PLAU
SCHEMBL1789555 0.82 CCR3 (0.49) MAPTHRH3CHRNA7ROCK2CHRM2
SCHEMBL4768264 0.81 HRH3 (0.50) NPC1RAB9AMAPTHRH3MELK
SCHEMBL4770147 0.81 HRH3 (0.46) NPC1RAB9AMAPTHRH3PLAU
SCHEMBL4765111 0.80 HRH3 (0.46) NPC1RAB9AMAPTHRH3MELK
SCHEMBL4768500 0.80 HRH3 (0.57) NPC1RAB9AHRH3PLAUTMPRSS2
SCHEMBL4768058 0.80 NPC1 (0.69) NPC1RAB9AMAPTHRH3MELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP claimed