SCHEMBL4768583

SCHEMBL4768583

O=C(Nc1ccc2c(c1)CCN(C1CCC1)CC2)c1cccc2ccccc12

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TMPRSS2 O15393 1/20 0.62
GAA P10253 1/20 0.52
NPC1 O15118 4/20 0.49
RAB9A P51151 3/20 0.49
TP53 P04637 1/20 0.49
MAPT P10636 1/20 0.49
NFKB1 P19838 1/20 0.49
HTT P42858 1/20 0.49
NFKB2 Q00653 1/20 0.49
RELA Q04206 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
DEGS1 O15121 1/20 0.48
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
RXFP1 Q9HBX9 1/20 0.47
ATM Q13315 1/20 0.47
ABCB1 P08183 1/20 0.47
ABCG2 Q9UNQ0 1/20 0.47
ALDH1A1 P00352 1/20 0.46
LMNA P02545 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4774158 0.93 TMPRSS2 (0.55) TMPRSS2GAANPC1RAB9ATP53
SCHEMBL4766059 0.85 KDM4E (0.50) TMPRSS2GAANPC1RAB9AMAPT
SCHEMBL4770555 0.85 NPC1 (0.51) GAANPC1RAB9ATP53MAPT
Hydrochloric Acid SCHEMBL4774323 0.85 KDM4E (0.49) TMPRSS2GAANPC1RAB9AMAPT
SCHEMBL4767370 0.83 MEN1 (0.58) GAANPC1RAB9ATP53MAPT
SCHEMBL4772757 0.82 HRH3 (0.52) NPC1RAB9ATP53MAPTNFKB1
SCHEMBL4768475 0.82 MEN1 (0.49) TMPRSS2GAANPC1RAB9ATP53
SCHEMBL4772451 0.82 TP53 (0.53) NPC1RAB9ATP53MAPTNFKB1
SCHEMBL4768212 0.82 NPC1 (0.58) NPC1RAB9ATP53MAPTSMN1; SMN2
SCHEMBL4774628 0.82 TMPRSS2 (0.61) TMPRSS2GAANPC1RAB9ATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP claimed