SCHEMBL4768694

SCHEMBL4768694

CC(C)(C)OC(=O)N1C[C@@H](O)[C@@H](Nc2cc(-c3cccnc3)nc(-c3ccccn3)n2)C1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIT P10721 2/20 0.44
GBA1 P04062 1/20 0.44
USP30 Q70CQ3 4/20 0.43
GPR119 Q8TDV5 2/20 0.41
ABL1 P00519 1/20 0.40
PDGFRB P09619 1/20 0.40
KDM1A O60341 1/20 0.39
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
TGFBR1 P36897 1/20 0.39
TGFBR2 P37173 1/20 0.39
BACE1 P56817 4/20 0.38
BACE2 Q9Y5Z0 1/20 0.38
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
DGAT2 Q96PD7 1/20 0.37
SYK P43405 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4772988 0.76 CYP2A6 (0.45) GBA1ABL1PDGFRBTGFBR1TGFBR2
SCHEMBL4775378 0.72 MERTK (0.52) CDK2SYK
SCHEMBL23416883 0.71 USP30 (0.42) KITGBA1USP30GPR119KDM1A
SCHEMBL4878463 0.71 SYK (0.47) GBA1CDK2SYK
SCHEMBL4773261 0.71 SYK (0.47) GBA1CDK2SYK
SCHEMBL2190446 0.69 USP30 (0.67) USP30GPR119DGAT2
SCHEMBL8736357 0.69 USP30 (0.51) USP30GPR119
SCHEMBL4773025 0.69 CYP2A6 (0.47)
SCHEMBL4775400 0.68 GBA1 (0.53) GBA1
SCHEMBL2238203 0.68 HDAC1 (0.42) TGFBR1TGFBR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed