SCHEMBL4772988

SCHEMBL4772988

O[C@H]1CCCC[C@@H]1Nc1cc(-c2cccnc2)nc(-c2ccccn2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
TP53 P04637 1/20 0.42
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.42
RAB9A P51151 1/20 0.42
GBA1 P04062 1/20 0.41
CYP19A1 P11511 1/20 0.40
CNR1 P21554 2/20 0.40
ADORA2A P29274 2/20 0.40
ADORA1 P30542 2/20 0.40
ADORA3 P0DMS8 1/20 0.40
EGFR P00533 1/20 0.40
GPR39 O43194 1/20 0.40
TGFBR1 P36897 1/20 0.40
TGFBR2 P37173 1/20 0.40
NPSR1 Q6W5P4 2/20 0.39
SLC2A1 P11166 2/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4773261 0.88 SYK (0.47) CYP2A6SMN1; SMN2NPC1TP53PKM
SCHEMBL4878463 0.88 SYK (0.47) CYP2A6SMN1; SMN2NPC1TP53PKM
SCHEMBL4775378 0.83 MERTK (0.52) CYP2A6SMN1; SMN2NPC1TP53PKM
SCHEMBL30085581 0.81 KMT2A (0.48) NPC1GBA1CNR1ADORA3NPSR1
SCHEMBL28895091 0.81 KMT2A (0.48) NPC1GBA1CNR1ADORA3NPSR1
SCHEMBL28895089 0.81 KMT2A (0.48) NPC1GBA1CNR1ADORA3NPSR1
SCHEMBL4773025 0.79 CYP2A6 (0.47) CYP2A6SMN1; SMN2NPC1TP53PKM
SCHEMBL4775007 0.77 ALDH1A1 (0.38) CYP2A6SMN1; SMN2NPC1TP53PKM
SCHEMBL4768694 0.76 KIT (0.44) GBA1TGFBR1TGFBR2ABL1PDGFRB
SCHEMBL4775400 0.76 GBA1 (0.53) CYP2A6SMN1; SMN2NPC1TP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed