SCHEMBL4775400

SCHEMBL4775400

c1ccc(-c2nc(NC3CCc4ccccc43)cc(-c3cccnc3)n2)nc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 2/20 0.53
PFKFB3 Q16875 11/20 0.46
CYP2A6 P11509 1/20 0.44
TSHR P16473 3/20 0.43
ALDH1A1 P00352 2/20 0.43
JAK2 O60674 2/20 0.42
JAK3 P52333 2/20 0.42
TP53 P04637 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
NPC1 O15118 1/20 0.41
PKM P14618 1/20 0.41
RAB9A P51151 1/20 0.41
NSD2 O96028 2/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
MAPK1 P28482 1/20 0.41
CASP1 P29466 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775378 0.78 MERTK (0.52) CYP2A6TSHRJAK2JAK3TP53
SCHEMBL4773025 0.78 CYP2A6 (0.47) CYP2A6TSHRJAK3TP53SMN1; SMN2
SCHEMBL4773261 0.76 SYK (0.47) GBA1CYP2A6TSHRJAK2JAK3
SCHEMBL4878463 0.76 SYK (0.47) GBA1CYP2A6TSHRJAK2JAK3
SCHEMBL4772988 0.76 CYP2A6 (0.45) GBA1CYP2A6TSHRTP53SMN1; SMN2
SCHEMBL4775007 0.72 ALDH1A1 (0.38) CYP2A6TSHRALDH1A1TP53SMN1; SMN2
SCHEMBL5691101 0.72 PDPK1 (0.53) TSHRALDH1A1JAK2JAK3TP53
SCHEMBL28657627 0.71 GBA1 (0.56) GBA1PFKFB3TSHRALDH1A1JAK2
SCHEMBL24589930 0.71 CYP2A6 (0.67) CYP2A6TSHRALDH1A1TP53SMN1; SMN2
SCHEMBL4775842 0.70 CYP3A4 (0.60) CYP2A6TSHRALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1878733-A1 Pyrimidine derivatives as ALK-5 inhibitors Novartis AG (CH) 2008-01-16 EP disclosed