SCHEMBL4769192

SCHEMBL4769192

O=[N+]([O-])c1ccc2[nH]c(C3CCCN3)nc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.50
ALDH1A1 P00352 3/20 0.45
RIPK1 Q13546 1/20 0.44
PARP1 P09874 5/20 0.43
TXN P10599 1/20 0.41
MAPT P10636 6/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
RAB9A P51151 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
POLB P06746 1/20 0.39
MAOB P27338 1/20 0.39
NOS1 P29475 1/20 0.39
LMNA P02545 1/20 0.39
NPC1 O15118 1/20 0.39
MMP2 P08253 1/20 0.39
MMP9 P14780 1/20 0.39
MMP8 P22894 1/20 0.39
CASP3 P42574 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769195 1.00 SCN10A (0.50) SCN10AALDH1A1RIPK1PARP1TXN
Hydrochloric Acid SCHEMBL30864304 0.99 SCN10A (0.49) SCN10AALDH1A1RIPK1PARP1TXN
Hydrochloric Acid SCHEMBL30204304 0.99 SCN10A (0.49) SCN10AALDH1A1RIPK1PARP1TXN
SCHEMBL23010726 0.83 RAB9A (0.53) ALDH1A1RIPK1TXNMAPTMEN1
SCHEMBL3576328 0.83 ALDH1A1 (0.52) ALDH1A1RIPK1TXNMAPTMEN1
SCHEMBL14447532 0.82 RAB9A (0.55) ALDH1A1RIPK1TXNMAPTMEN1
SCHEMBL7970193 0.81 ALDH1A1 (0.48) ALDH1A1RIPK1PARP1TXNMAPT
SCHEMBL12509313 0.80 SCN10A (0.58) SCN10APARP1
SCHEMBL1645792 0.79 SCN10A (0.56) SCN10APARP1
SCHEMBL9605019 0.79 SCN10A (0.56) SCN10APARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1973898-A1 PDF INHIBITORS Novartis AG (CH) 2008-10-01 EP disclosed
WO-2007077186-A1 PDF INHIBITORS NOVARTIS AG (CH) 2007-07-12 WO disclosed