SCHEMBL4771053

SCHEMBL4771053

CC(C)C[C@](CNCCCCNS(=O)(=O)c1ccc(Cl)cc1Cl)(NC(=O)O)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.39
TRPV4 Q9HBA0 7/20 0.39
GAA P10253 1/20 0.38
CNR1 P21554 2/20 0.37
CNR2 P34972 2/20 0.37
ATM Q13315 1/20 0.36
FABP4 P15090 1/20 0.36
ALDH1A1 P00352 1/20 0.35
ITGA1 P56199 1/20 0.35
TBXAS1 P24557 1/20 0.35
MEN1 O00255 1/20 0.34
TSHR P16473 1/20 0.34
KMT2A Q03164 1/20 0.34
APP P05067 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135486 0.76 CCR1 (0.42) CCR1TRPV4GAACNR1CNR2
SCHEMBL4768147 0.75 CCR1 (0.42) CCR1TRPV4GAACNR1CNR2
SCHEMBL4140000 0.74 CCR1 (0.47) CCR1TRPV4GAACNR1CNR2
SCHEMBL13872499 0.70 AAK1 (0.46) CCR1TRPV4GAAATMALDH1A1
SCHEMBL4975544 0.70 MAPT (0.39) CCR1TRPV4ATMALDH1A1MEN1
SCHEMBL13872450 0.69 IDO1 (0.47) CCR1TRPV4GAACNR1CNR2
SCHEMBL14605764 0.69 TRPV4 (0.43) CCR1TRPV4GAACNR1ATM
SCHEMBL14606011 0.69 CCR1 (0.39) CCR1TRPV4GAACNR1CNR2
SCHEMBL4132204 0.69 MAPK1 (0.45) CCR1TRPV4CNR1ATMFABP4
SCHEMBL4132203 0.69 MAPK1 (0.45) CCR1TRPV4CNR1ATMFABP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed