SCHEMBL4768147

SCHEMBL4768147

CC(C)(C)C(CNCCCCNS(=O)(=O)c1ccc(Cl)cc1Cl)NC(=O)O

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 1/20 0.42
TRPV4 Q9HBA0 7/20 0.42
GAA P10253 1/20 0.41
CNR1 P21554 2/20 0.40
CNR2 P34972 2/20 0.40
ITGAV P06756 1/20 0.40
FABP4 P15090 2/20 0.39
ITGA1 P56199 2/20 0.38
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPK1 P28482 1/20 0.37
ATM Q13315 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4135486 0.84 CCR1 (0.42) CCR1TRPV4GAACNR1CNR2
SCHEMBL4773183 0.80 GAA (0.40) CCR1TRPV4GAACNR1CNR2
SCHEMBL4140000 0.78 CCR1 (0.47) CCR1TRPV4GAACNR1CNR2
SCHEMBL14605764 0.77 TRPV4 (0.43) CCR1TRPV4GAACNR1FABP4
SCHEMBL13872499 0.76 AAK1 (0.46) CCR1TRPV4GAAKDM4EALDH1A1
SCHEMBL4127274 0.76 TRPV4 (0.47) CCR1TRPV4GAAALDH1A1
SCHEMBL3913649 0.76 ITGA1 (0.43) CCR1TRPV4CNR2ITGAVITGA1
SCHEMBL14606011 0.75 CCR1 (0.39) CCR1TRPV4GAACNR1CNR2
SCHEMBL4771053 0.75 CCR1 (0.39) CCR1TRPV4GAACNR1CNR2
SCHEMBL4132204 0.75 MAPK1 (0.45) CCR1TRPV4CNR1FABP4ITGA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940785-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007030761-A2 ACYCLIC 1,4-DIAMINES AND USES THEREOF SMITHKLINE BEECHAM CORPORATION (US) 2007-03-15 WO disclosed