SCHEMBL4771056

SCHEMBL4771056

CNc1ccccc1N(C=O)CCN(C=O)c1ccc(N(Cc2cccc(Cl)c2Cl)S(C)(=O)=O)cc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.37
ALDH1A1 P00352 2/20 0.36
MAPT P10636 2/20 0.35
NR3C1 P04150 1/20 0.35
LMNA P02545 2/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
GLA P06280 1/20 0.35
CYP2D6 P10635 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MAPK1 P28482 1/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
RECQL P46063 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
POLB P06746 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4768018 0.83 ALDH1A1 (0.43) GAAALDH1A1MAPTLMNANPSR1
SCHEMBL4777347 0.78 NR1H4 (0.39) GAAALDH1A1MAPTLMNACYP1A2
SCHEMBL4776590 0.78 GAA (0.42) GAAALDH1A1MAPTLMNANPSR1
SCHEMBL4777561 0.77 GAA (0.36) GAAALDH1A1MAPTLMNACYP1A2
SCHEMBL4777314 0.77 GAA (0.38) GAAALDH1A1MAPTLMNACYP1A2
SCHEMBL4771365 0.76 GAA (0.37) GAAALDH1A1MAPTLMNACYP1A2
SCHEMBL5571819 0.76 SLC6A4 (0.42) GAAALDH1A1MAPTLMNACYP1A2
SCHEMBL4775060 0.75 GAA (0.39) GAAALDH1A1MAPTLMNANPSR1
SCHEMBL4775247 0.74 GAA (0.48) GAAALDH1A1MAPTLMNANPSR1
SCHEMBL4768047 0.74 REN (0.41) GAAALDH1A1MAPTLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed