SCHEMBL4771531

SCHEMBL4771531

CC(C)Cn1c(/C=C/c2cnn(Cc3ccccc3F)c2)c([N+](=O)[O-])c(=O)n(CCc2ccccc2)c1=O

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 9/20 0.38
ADORA2A P29274 7/20 0.38
ADORA1 P30542 7/20 0.38
ADORA3 P0DMS8 4/20 0.38
TP53 P04637 2/20 0.38
GNRHR P30968 1/20 0.34
TSHR P16473 1/20 0.34
MAPT P10636 2/20 0.34
GAA P10253 1/20 0.34
ALDH1A1 P00352 1/20 0.33
PKM P14618 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
LMNA P02545 1/20 0.33
MAPK1 P28482 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC2 Q92769 1/20 0.33
THRB P10828 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771549 1.00 ADORA2B (0.38) ADORA2BADORA2AADORA1ADORA3TP53
SCHEMBL4765722 0.93 TP53 (0.41) ADORA2BADORA2AADORA1TP53TSHR
SCHEMBL4765708 0.93 TP53 (0.41) ADORA2BADORA2AADORA1TP53TSHR
SCHEMBL4762309 0.93 ADORA2B (0.39) ADORA2BADORA2AADORA1ADORA3GNRHR
SCHEMBL4762305 0.93 ADORA2B (0.39) ADORA2BADORA2AADORA1ADORA3GNRHR
SCHEMBL4764018 0.91 ADORA2B (0.41) ADORA2BADORA2AADORA1ADORA3GNRHR
SCHEMBL4764008 0.91 ADORA2B (0.41) ADORA2BADORA2AADORA1ADORA3GNRHR
SCHEMBL4767738 0.88 ADORA2B (0.41) ADORA2BADORA2AADORA1ADORA3MAPT
SCHEMBL4767746 0.88 ADORA2B (0.41) ADORA2BADORA2AADORA1ADORA3MAPT
SCHEMBL4771540 0.86 ADORA2B (0.40) ADORA2BADORA2AADORA1ADORA3GNRHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678181-B1 A2B ADENOSINE RECEPTOR ANTAGONISTS CV THERAPEUTICS INC (US) 2008-12-31 EP disclosed