SCHEMBL4771677

SCHEMBL4771677

CCCS(=O)(=O)c1ccc(CC2CCNCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.50
MLNR O43193 2/20 0.45
NMT1 P30419 4/20 0.39
ITGB3 P05106 1/20 0.38
ITGA2B P08514 1/20 0.38
SLC6A4 P31645 2/20 0.38
PNMT P11086 1/20 0.38
HTR6 P50406 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
PSIP1 O75475 1/20 0.37
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4770307 0.92 MLNR (0.49) GBA1MLNRNMT1ITGB3ITGA2B
SCHEMBL4777240 0.89 GBA1 (0.54) GBA1MLNRNMT1SLC6A4HTR6
Hydrochloric Acid SCHEMBL4773264 0.88 GBA1 (0.53) GBA1MLNRNMT1SLC6A4HTR6
SCHEMBL4775645 0.85 GBA1 (0.44) GBA1MLNRNMT1ITGB3ITGA2B
SCHEMBL3037834 0.81 GBA1 (0.56) GBA1NMT1SLC6A4SMN1; SMN2
SCHEMBL4771338 0.81 GBA1 (0.49) GBA1MLNRNMT1SLC6A4SMN1; SMN2
Hydrochloric Acid SCHEMBL4768496 0.81 HTR2C (0.52) GBA1NMT1PNMTSMN1; SMN2ALDH1A1
Hydrochloric Acid SCHEMBL3034504 0.80 GBA1 (0.54) GBA1NMT1SLC6A4SMN1; SMN2
SCHEMBL28963842 0.79 MLNR (0.41) GBA1MLNRNMT1ITGB3ITGA2B
SCHEMBL25145663 0.78 GBA1 (0.56) GBA1NMT1SLC6A4SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists TOBIRA THERAPEUTICS, INC. 2003-06-19 US disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed
EP-1220842-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-10 EP disclosed
WO-2001025200-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists CCR5, CCR1, CCR3 GBA1 2987/4885MLNR 1474/4885NMT1 661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.