SCHEMBL4775645

SCHEMBL4775645

CCOCCS(=O)(=O)c1ccc(CC2CCNCC2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.44
SLC6A4 P31645 3/20 0.42
LOX P28300 1/20 0.42
MLNR O43193 2/20 0.39
HTR6 P50406 1/20 0.36
KCNH2 Q12809 1/20 0.36
NMT1 P30419 4/20 0.36
ALDH1A1 P00352 1/20 0.36
ITGB3 P05106 3/20 0.35
ITGA2B P08514 3/20 0.35
ITGAV P06756 1/20 0.35
CHRM2 P08172 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771677 0.85 GBA1 (0.50) GBA1SLC6A4MLNRHTR6NMT1
SCHEMBL4777240 0.83 GBA1 (0.54) GBA1SLC6A4MLNRHTR6NMT1
SCHEMBL4770307 0.83 MLNR (0.49) GBA1SLC6A4MLNRHTR6KCNH2
Hydrochloric Acid SCHEMBL4773264 0.82 GBA1 (0.53) GBA1SLC6A4MLNRHTR6NMT1
SCHEMBL4779005 0.81 ALDH1A1 (0.51) ALDH1A1
SCHEMBL7513018 0.79 ALDH1A1 (0.39) LOXKCNH2ALDH1A1
SCHEMBL3037834 0.76 GBA1 (0.56) GBA1SLC6A4NMT1
SCHEMBL4771338 0.76 GBA1 (0.49) GBA1SLC6A4MLNRNMT1
Hydrochloric Acid SCHEMBL3034504 0.75 GBA1 (0.54) GBA1SLC6A4NMT1
SCHEMBL25145663 0.73 GBA1 (0.56) GBA1SLC6A4KCNH2NMT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists TOBIRA THERAPEUTICS, INC. 2003-06-19 US disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed
EP-1220842-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-10 EP disclosed
WO-2001025200-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists CCR5, CCR1, CCR3 GBA1 2987/4885SLC6A4 559/4885LOX 2150/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.