SCHEMBL4777240

SCHEMBL4777240

CCS(=O)(=O)c1ccc(CC2CCNCC2)cc1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GBA1 P04062 1/20 0.54
PSIP1 O75475 2/20 0.47
MLNR O43193 2/20 0.42
RORC P51449 3/20 0.41
GAA P10253 2/20 0.41
SLC6A4 P31645 2/20 0.40
HTR6 P50406 1/20 0.39
NMT1 P30419 2/20 0.39
CNR2 P34972 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4773264 0.98 GBA1 (0.53) GBA1PSIP1MLNRRORCGAA
SCHEMBL4771677 0.89 GBA1 (0.50) GBA1PSIP1MLNRSLC6A4HTR6
SCHEMBL4770307 0.87 MLNR (0.49) GBA1MLNRSLC6A4HTR6NMT1
SCHEMBL3037834 0.85 GBA1 (0.56) GBA1RORCGAASLC6A4NMT1
SCHEMBL4771338 0.85 GBA1 (0.49) GBA1MLNRGAASLC6A4NMT1
Hydrochloric Acid SCHEMBL3034504 0.84 GBA1 (0.54) GBA1RORCGAASLC6A4NMT1
SCHEMBL4775645 0.83 GBA1 (0.44) GBA1MLNRSLC6A4HTR6NMT1
SCHEMBL25145663 0.82 GBA1 (0.56) GBA1GAASLC6A4NMT1CNR2
SCHEMBL27917814 0.82 GBA1 (0.56) GBA1HTTSMN1; SMN2
SCHEMBL4768607 0.82 HTT (0.50) GBA1GAANMT1TSHRHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7348324-B2 Cyclic amine compounds as CCR5 antagonists TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-03-25 US disclosed
EP-1886994-A1 Cyclic amine compounds as CCR5 antagonists Takeda Pharmaceutical Company Limited (JP) 2008-02-13 EP disclosed
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists TOBIRA THERAPEUTICS, INC. 2003-06-19 US disclosed
US-6562978-B1 N-(3-(4-(4-(Aminocarbonyl)benzyl)-1-piperidinyl)propyl)-N-(3, 4-dichlorophenyl)-1-(methylsulfonyl)-4-piperidinecarboxamide or a salt thereof for treatment of AIDS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-05-13 US disclosed
CN-1390201-A cyclic amine compounds as CCR5 antagonists TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-01-08 CN disclosed
EP-1220842-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS Takeda Chemical Industries, Ltd. (JP) 2002-07-10 EP disclosed
WO-2001025200-A1 CYCLIC AMINE COMPOUNDS AS CCR5 ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030114443-A1 Cyclic amine compounds as CCR5 antagonists CCR5, CCR1, CCR3 GBA1 2987/4885PSIP1 4443/4885MLNR 1474/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.