SCHEMBL4773616

SCHEMBL4773616

CCOC(=O)c1cn(-c2ccccc2)c2nc(N(CC)C3CCCN3)ncc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 6/20 0.43
PDE4B Q07343 1/20 0.37
ALDH1A1 P00352 3/20 0.36
ATM Q13315 1/20 0.36
TSHR P16473 2/20 0.36
MAPK1 P28482 1/20 0.36
MAPT P10636 2/20 0.36
PDE4A P27815 1/20 0.36
KCNH2 Q12809 1/20 0.36
ELANE P08246 1/20 0.36
PIM1 P11309 1/20 0.36
IRAK1 P51617 1/20 0.36
CAMK2B Q13554 1/20 0.36
CAMK2G Q13555 1/20 0.36
CAMK2D Q13557 1/20 0.36
PIM3 Q86V86 1/20 0.36
KDM4E B2RXH2 2/20 0.36
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769014 0.98 CSF1R (0.42) CSF1RPDE4BALDH1A1ATMTSHR
SCHEMBL4775340 0.90 CSF1R (0.48) CSF1RPDE4AKCNH2
SCHEMBL4768393 0.87 CSF1R (0.47) CSF1RPDE4ACCNA2CDK2CCNA1
SCHEMBL4775457 0.86 CSF1R (0.57) CSF1R
SCHEMBL4771887 0.86 CSF1R (0.40) CSF1RMAPK1PDE4AKCNH2KDM4E
SCHEMBL4775791 0.82 CSF1R (0.39) CSF1RPDE4BALDH1A1ATMTSHR
SCHEMBL4572926 0.76 CSF1R (0.53) CSF1R
SCHEMBL4773660 0.75 CSF1R (0.56) CSF1R
SCHEMBL16088470 0.74 CSF1R (0.44) CSF1RALDH1A1TSHRMAPK1MAPT
SCHEMBL28537798 0.74 CSF1R (0.62) CSF1RPDE4BMAPTNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945637-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA N.V. (BE) 2008-07-23 EP disclosed
WO-2007033137-A1 5-OXO-5,8-DIHYDRO-PYRIDO-PYRIMIDINES AS INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA, N.V. (BE) 2007-03-22 WO disclosed