SCHEMBL4774558

SCHEMBL4774558

Cc1cc(C)n2nc(C(=O)Nc3ccc4c(c3)CCN(C3CCC3)CC4)cc2n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.59
RAB9A P51151 6/20 0.59
SMN1; SMN2 Q16637 6/20 0.59
ALDH1A1 P00352 6/20 0.59
MAPT P10636 6/20 0.59
KDM4E B2RXH2 6/20 0.59
HPGD P15428 4/20 0.54
HSD17B10 Q99714 3/20 0.54
TP53 P04637 3/20 0.54
TSHR P16473 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
KMT2A Q03164 4/20 0.53
MEN1 O00255 2/20 0.53
USP2 O75604 2/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
HRH3 Q9Y5N1 6/20 0.45
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
RELA Q04206 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL4775303 0.94 ALDH1A1 (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4767869 0.82 HRH3 (0.49) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4776972 0.80 AURKA (0.54) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL4767326 0.79 RAB9A (0.71) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4777120 0.79 NPY5R (0.54) NPC1RAB9ASMN1; SMN2MAPTTP53
SCHEMBL4772665 0.77 HRH3 (0.52) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4770392 0.77 HRH3 (0.59) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4770662 0.77 MEN1 (0.57) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4767967 0.77 HRH3 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT
SCHEMBL4774177 0.75 HRH3 (0.69) NPC1RAB9ASMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1713778-B1 BENZAZEPINE DERIVATIVES AS HISTAMINE H3 ANTAGONISTS GLAXO GROUP LTD (GB) 2008-01-16 EP claimed