SCHEMBL4775829

SCHEMBL4775829

CC1(C)CNCc2c1nn(C(=O)O)c2NC(=O)c1ccccc1[N+](=O)[O-]

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
HTT P42858 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
GAA P10253 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
LMNA P02545 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4D Q08499 1/20 0.41
ALDH1A1 P00352 2/20 0.39
HPGD P15428 1/20 0.39
NPC1 O15118 1/20 0.39
MAPK1 P28482 1/20 0.39
ABCG2 Q9UNQ0 1/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2677894 0.88 ALDH1A1 (0.46) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL2677890 0.88 ALDH1A1 (0.46) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL4424639 0.76 ALDH1A1 (0.48) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL4424633 0.75 ALDH1A1 (0.48) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL2677500 0.75 MAPT (0.36) KDM4ECYP3A4CYP2C19HTTSMN1; SMN2
SCHEMBL2678711 0.73 L3MBTL1 (0.36) SMN1; SMN2GAALMNAALDH1A1MAPK1
SCHEMBL2679062 0.73 MAPT (0.40) CYP1A2SMN1; SMN2LMNAALDH1A1NPC1
Hydrochloric Acid SCHEMBL2678981 0.73 SIRT6 (0.40) SMN1; SMN2LMNAALDH1A1MAPK1MAPT
Hydrochloric Acid SCHEMBL2678708 0.73 L3MBTL1 (0.35) SMN1; SMN2GAALMNAALDH1A1MAPK1
SCHEMBL4532323 0.71 KMT2A (0.42) KDM4EHTTSMN1; SMN2GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968976-A1 SUBSTITUTED PYRAZOLO [4,3-C] PYRIDINE DERIVATIVES ACTIVE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.r.l. (IT) 2008-09-17 EP disclosed
WO-2007068619-A1 SUBSTITUTED PYRAZOLO [4,3-C] PYRIDINE DERIVATIVES ACTIVE AS KINASE INHIBITORS NERVIANO MEDICAL SCIENCES S.R.L. (IT) 2007-06-21 WO disclosed