SCHEMBL4775874

SCHEMBL4775874

O=C1c2ccccc2OC1F

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.45
KDR P35968 1/20 0.45
CYP19A1 P11511 7/20 0.43
MAOB P27338 3/20 0.43
ADORA3 P0DMS8 2/20 0.43
AR P10275 2/20 0.43
MEN1 O00255 2/20 0.43
POLB P06746 2/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
STK17B O94768 1/20 0.42
PARP1 P09874 1/20 0.40
S100A4 P26447 1/20 0.38
HSD11B1 P28845 1/20 0.38
AKR1C3 P42330 1/20 0.38
PKM P14618 1/20 0.38
TSHR P16473 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548145 0.76 RET (0.46) RETKDRCYP19A1MAOBADORA3
SCHEMBL69430 0.74 PARP1 (0.48) RETKDRCYP19A1MAOBADORA3
SCHEMBL1429502 0.74 STK17B (0.46) RETKDRCYP19A1MAOBADORA3
SCHEMBL69727 0.74 RET (0.53) RETKDRCYP19A1MAOBADORA3
SCHEMBL29441433 0.72 MEN1 (0.52) RETKDRCYP19A1MAOBADORA3
SCHEMBL28875665 0.72 MEN1 (0.52) RETKDRCYP19A1MAOBADORA3
SCHEMBL9837501 0.72 RET (0.41) RETKDRCYP19A1MAOBADORA3
SCHEMBL10513412 0.71 STK17B (0.51) RETKDRCYP19A1MAOBADORA3
SCHEMBL92288 0.71 ESR1 (0.45) RETKDRCYP19A1MAOBADORA3
SCHEMBL9434848 0.71 ESR1 (0.45) RETKDRCYP19A1MAOBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109942556-A Pyrimidinone compound and its application 上海青煜医药科技有限公司 2019-06-28 CN disclosed
WO-2008084067-A2 PHARMACEUTICALLY ACTIVE DIHYDROBENZOFURANE-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES NYCOMED GMBH (DE) 2008-07-17 WO disclosed
EP-1874772-A1 PURINE AND IMIDAZOPYRIDINE DERIVATIVES FOR IMMUNOSUPPRESSION PHARMACOPEIA, INC. (US) 2008-01-09 EP disclosed
WO-2006108103-A1 PURINE AND IMIDAZOPYRIDINE DERIVATIVES FOR IMMUNOSUPPRESSION PHARMACOPEIA, INC. (US) 2006-10-12 WO disclosed