SCHEMBL4776309

SCHEMBL4776309

Cc1ccc(Cl)cc1N1CCN(C(c2ccc(C(F)(F)F)cc2)C(N)C=O)CC1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.42
ALDH1A1 P00352 3/20 0.41
MC4R P32245 11/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MCOLN3 Q8TDD5 1/20 0.40
USP2 O75604 2/20 0.39
LMNA P02545 2/20 0.39
TSHR P16473 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
RPS6KB1 P23443 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4771297 0.80 NPSR1 (0.46) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL4776952 0.79 LMNA (0.46) NPSR1ALDH1A1MC4RMEN1KMT2A
SCHEMBL4779189 0.78 NPSR1 (0.43) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL4776587 0.77 KDM4E (0.45) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL4773595 0.75 ALDH1A1 (0.43) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL4770304 0.73 NPSR1 (0.39) NPSR1ALDH1A1MEN1KMT2AMCOLN3
SCHEMBL23549955 0.71 USP2 (0.55) NPSR1ALDH1A1MC4RMEN1KMT2A
SCHEMBL19403828 0.71 USP2 (0.55) NPSR1ALDH1A1MC4RMEN1KMT2A
SCHEMBL4778512 0.71 MC4R (0.58) ALDH1A1MC4RMEN1KMT2AUSP2
SCHEMBL19403735 0.70 NPSR1 (0.45) NPSR1ALDH1A1MC4RMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996550-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES Novartis AG (CH) 2008-12-03 EP disclosed
WO-2007038459-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES NOVARTIS AG (CH) 2007-04-05 WO disclosed