SCHEMBL4776444

SCHEMBL4776444

COc1ccc(S(=O)(=O)n2cc(C=O)c3cc(Br)ccc32)c(Br)c1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.46
CYP3A4 P08684 2/20 0.46
ADRA2A P08913 2/20 0.46
CYP2D6 P10635 2/20 0.46
ADRA2C P18825 2/20 0.46
CYP2C19 P33261 2/20 0.46
HTR2A P28223 1/20 0.46
ALDH1A1 P00352 1/20 0.44
KDM4E B2RXH2 1/20 0.39
UBE2N P61088 1/20 0.39
PDK1 Q15118 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4769905 0.94 HTR6 (0.50) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4773184 0.89 HTR6 (0.44) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4774296 0.87 KDM4E (0.54) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4772681 0.86 HTR6 (0.60) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4778090 0.86 KDM4E (0.52) HTR6CYP3A4CYP2D6ALDH1A1KDM4E
SCHEMBL4774289 0.85 HTR6 (0.47) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4778240 0.84 HTR6 (0.59) HTR6CYP3A4CYP2D6HTR2AALDH1A1
SCHEMBL949730 0.82 HTR6 (0.58) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL4770622 0.81 HTR6 (0.54) HTR6CYP3A4ADRA2ACYP2D6ADRA2C
SCHEMBL945974 0.81 HTR6 (0.54) HTR6CYP3A4ADRA2ACYP2D6ADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581492-B1 N-ARYLSULFONYL-3-SUBSTITUTED INDOLES HAVING SEROTONIN RECEPTOR AFFINITY, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM SUVEN LIFE SCIENCES LTD (IN) 2008-07-16 EP disclosed