SCHEMBL4776564

SCHEMBL4776564

N=C(N)Nc1ccc(-c2cc(Cc3ccc4ccccc4c3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.37
SPHK1 Q9NYA1 8/20 0.35
EPHX1 P07099 2/20 0.34
BDKRB2 P30411 1/20 0.34
SPHK2 Q9NRA0 7/20 0.34
CCNB2 O95067 1/20 0.33
CCNE2 O96020 1/20 0.33
CDK1 P06493 1/20 0.33
CCNB1 P14635 1/20 0.33
CCNA2 P20248 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
CDK5 Q00535 1/20 0.33
CDK5R1 Q15078 1/20 0.33
CCNB3 Q8WWL7 1/20 0.33
BACE1 P56817 1/20 0.33
METAP2 P50579 1/20 0.32
METAP1 P53582 1/20 0.32
PDE5A O76074 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780443 0.83 PDE5A (0.38) SPHK1PDE5A
SCHEMBL4776487 0.83 PDE5A (0.38) SPHK1PDE5A
SCHEMBL4796379 0.83 PDE5A (0.38) SPHK1PDE5A
SCHEMBL4780605 0.74 BRAF (0.38) SPHK2METAP2PDE5A
SCHEMBL14303801 0.72 KDM4E (0.40) EPHX1
SCHEMBL4776439 0.70 SPHK1 (0.35) SPHK1EPHX1PDE5A
SCHEMBL4780429 0.70 MOK (0.42) EPHX1
SCHEMBL4796206 0.69 SPHK1 (0.37) SPHK1
SCHEMBL4779379 0.67 SPHK1 (0.34) SPHK1PDE5A
SCHEMBL4778365 0.66 PDE5A (0.40) EPHX1PDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed