SCHEMBL4776439

SCHEMBL4776439

N=C(N)Nc1ccc(Oc2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SPHK1 Q9NYA1 10/20 0.35
MAPT P10636 3/20 0.35
ALOX12 P18054 3/20 0.35
HTT P42858 3/20 0.35
ALDH1A1 P00352 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 2/20 0.34
EPHX1 P07099 1/20 0.34
TP53 P04637 1/20 0.34
OPRM1 P35372 2/20 0.34
MCHR1 Q99705 2/20 0.33
PDE5A O76074 1/20 0.33
NAPEPLD Q6IQ20 1/20 0.33
MCHR2 Q969V1 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780443 0.85 PDE5A (0.38) SPHK1ALDH1A1PDE5A
SCHEMBL4796379 0.85 PDE5A (0.38) SPHK1ALDH1A1PDE5A
SCHEMBL4776487 0.85 PDE5A (0.38) SPHK1ALDH1A1PDE5A
SCHEMBL4774683 0.85 NOS3 (0.39) MAPTALDH1A1LMNAMCHR1PDE5A
SCHEMBL4780605 0.80 BRAF (0.38) MAPTALDH1A1SMN1; SMN2LMNAPDE5A
SCHEMBL4794914 0.79 ADRA2A (0.45)
SCHEMBL4774580 0.79 GRIN2B (0.40) MAPTHTTALDH1A1LMNAEPHX1
SCHEMBL14303801 0.74 KDM4E (0.40) MAPTALDH1A1SMN1; SMN2EPHX1
SCHEMBL4780429 0.72 MOK (0.42) MAPTALDH1A1SMN1; SMN2EPHX1
SCHEMBL4774754 0.72 PDE5A (0.41) HTTEPHX1OPRM1PDE5AOPRD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed