SCHEMBL4780443

SCHEMBL4780443

N=C(N)Nc1ccc(-c2cc(CCCc3ccccc3)nc(C3CCCCC3)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.38
SPHK1 Q9NYA1 10/20 0.37
VCP P55072 1/20 0.36
ADORA1 P30542 2/20 0.34
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
DHODH Q02127 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
ATR Q13535 1/20 0.33
EPHX2 P34913 1/20 0.33
ADORA2A P29274 1/20 0.33
NAMPT P43490 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776487 1.00 PDE5A (0.38) PDE5ASPHK1VCPADORA1NOS3
SCHEMBL4796379 1.00 PDE5A (0.38) PDE5ASPHK1VCPADORA1NOS3
SCHEMBL4780605 0.90 BRAF (0.38) PDE5AADORA1NOS3NOS1NOS2
SCHEMBL14303801 0.88 KDM4E (0.40) KDM4EALDH1A1EPHX2
SCHEMBL4780429 0.87 MOK (0.42) ADORA1KDM4EALDH1A1EPHX2
SCHEMBL4776439 0.85 SPHK1 (0.35) PDE5ASPHK1ALDH1A1
SCHEMBL4796206 0.85 SPHK1 (0.37) SPHK1VCPNOS3NOS1NOS2
SCHEMBL4774100 0.83 NOS3 (0.42) PDE5AVCPADORA1NOS3NOS1
SCHEMBL4776564 0.83 TACR1 (0.37) PDE5ASPHK1
SCHEMBL4778365 0.82 PDE5A (0.40) PDE5AVCPADORA1NOS3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed
WO-2008009963-A2 PYRIMIDINE DERIVATIVES AS MODULATORS OF PARATHYROID HORMONE RECEPTORS JAMES BLACK FOUNDATION LIMITED (GB) 2008-01-24 WO disclosed