SCHEMBL4776685

SCHEMBL4776685

O=C(c1ccccc1)C1CN(CCCO)CC(C(=O)c2ccccc2)C1c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.43
KMT2A Q03164 3/20 0.41
MEN1 O00255 1/20 0.41
KCNH2 Q12809 1/20 0.41
TSHR P16473 1/20 0.40
ALDH1A1 P00352 3/20 0.39
LMNA P02545 2/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
HTR2A P28223 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RECQL P46063 1/20 0.38
SLC18A3 Q16572 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4020589 1.00 RORC (0.43) RORCKMT2AMEN1KCNH2TSHR
SCHEMBL4026119 0.92 SLC18A3 (0.45) RORCKMT2AMEN1KCNH2ALDH1A1
SCHEMBL4024282 0.92 SLC18A3 (0.45) RORCKMT2AMEN1KCNH2ALDH1A1
SCHEMBL4772340 0.84 KMT2A (0.48) RORCKMT2AMEN1KCNH2ALDH1A1
SCHEMBL4019373 0.84 KMT2A (0.46) RORCKMT2AMEN1ALDH1A1LMNA
SCHEMBL4026548 0.84 KMT2A (0.46) RORCKMT2AMEN1ALDH1A1LMNA
SCHEMBL4019381 0.84 KMT2A (0.46) RORCKMT2AMEN1ALDH1A1LMNA
SCHEMBL4772338 0.81 HRH3 (0.45) RORCKMT2AMEN1KCNH2ALDH1A1
SCHEMBL4021931 0.81 ALDH1A1 (0.55) KMT2AMEN1TSHRALDH1A1LMNA
SCHEMBL4774189 0.81 NTRK1 (0.43) RORCKMT2AMEN1ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1962846-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-09-03 EP disclosed
WO-2007059323-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-24 WO disclosed