SCHEMBL4776876

SCHEMBL4776876

CC(CCc1nc(=O)c2ncn(CC(F)F)c2n1-c1ccc(F)cc1)C(F)(F)F

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
RAB9A P51151 1/20 0.33
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4284448 0.93 NPC1 (0.34) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4769839 0.87 NPC1 (0.33) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4425849 0.84 NPC1 (0.37) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4529223 0.78 HKDC1 (0.40) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4512742 0.77 CNR1 (0.39) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4521064 0.75 HKDC1 (0.40) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4510793 0.72 HKDC1 (0.39) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4776782 0.70 CDK1 (0.33) NPC1LMNAHPGDTSHRRAB9A
SCHEMBL4357095 0.69 MAT2A (0.38) NPC1ALDH1A1LMNAHPGDTSHR
SCHEMBL4768907 0.69 SMN1; SMN2 (0.34) NPC1ALDH1A1LMNAHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881988-A1 2,3-SUBSTITUTED FUSED BICYCLIC PYRIMIDIN-4(3H)-ONES MODULATING THE FUNCTION OF THE VANILLOID-1 RECEPTOR (VR1) MERCK SHARP & DOHME LTD. (GB) 2008-01-30 EP disclosed
WO-2006122200-A1 2,3-SUBSTITUTED FUSED BICYCLIC PYRIMIDIN-4(3H)-ONES MODULATING THE FUNCTION OF THE VANILLOID-1 RECEPTOR (VR1) MERCK SHARP & DOHME LIMITED (GB) 2006-11-16 WO disclosed