SCHEMBL4776918

SCHEMBL4776918

CN(C(=O)c1ccc(N(Cc2cccc(Cl)c2Cl)C(=O)O)cc1)c1ccc(C(F)(F)F)nc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 2/20 0.41
GPBAR1 Q8TDU6 8/20 0.40
P2RX7 Q99572 3/20 0.39
OXTR P30559 1/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.37
NR1H3 Q13133 2/20 0.37
NR1H2 P55055 1/20 0.37
PDK1 Q15118 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
SLC6A2 P23975 1/20 0.36
SLC6A4 P31645 1/20 0.36
CYP2C19 P33261 1/20 0.36
SLC6A3 Q01959 1/20 0.36
KCNH2 Q12809 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4767615 0.93 NR1H3 (0.41) TRPM8GPBAR1P2RX7OXTRPTGDR2
SCHEMBL4777521 0.90 GPBAR1 (0.42) TRPM8GPBAR1P2RX7OXTR
SCHEMBL4771001 0.78 ALDH1A1 (0.36) TRPM8GPBAR1P2RX7OXTR
SCHEMBL4793541 0.78 KCNH2 (0.42) TRPM8P2RX7PDK1CYP1A2CYP3A4
SCHEMBL4767613 0.78 NAMPT (0.46) P2RX7
SCHEMBL4767893 0.77 TRPM8 (0.37) TRPM8GPBAR1OXTRCYP1A2CYP3A4
SCHEMBL4771084 0.77 GPBAR1 (0.37) TRPM8GPBAR1P2RX7OXTR
SCHEMBL4777432 0.77 TRPM8 (0.37) TRPM8GPBAR1P2RX7OXTR
SCHEMBL4777539 0.76 GPBAR1 (0.36) TRPM8GPBAR1P2RX7OXTR
SCHEMBL4777438 0.76 TRPM8 (0.36) TRPM8GPBAR1OXTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP claimed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO claimed