SCHEMBL4777038

SCHEMBL4777038

CCCOc1ccc(-c2ccc(C(C(N)C=O)N3CCN(C)CC3)s2)c(C)c1

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 3/20 0.32
MAPK1 P28482 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
ESR1 P03372 4/20 0.31
ESR2 Q92731 4/20 0.31
ACACB O00763 3/20 0.31
ACACA Q13085 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
HRH3 Q9Y5N1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4775579 0.73 MEN1 (0.41) ACACBACACAKDM4EALDH1A1MEN1
SCHEMBL3652692 0.60 REN (0.44) KDM4EALDH1A1
SCHEMBL5599357 0.59 ACACB (0.63) SMN1; SMN2ACACBACACAKDM4EALDH1A1
SCHEMBL3725442 0.58 ERN1 (0.48) MAPK1KDM4EALDH1A1TSHRMEN1
SCHEMBL15859178 0.57 ALDH1A1 (0.40) SMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL9098174 0.57 INPPL1 (0.42) MAPK1KDM4EALDH1A1MEN1KMT2A
SCHEMBL469900 0.56 DRD2 (0.53) SMN1; SMN2ACACBACACAKDM4EMEN1
SCHEMBL20772370 0.56 HSD17B2 (0.43) SMN1; SMN2KDM4EALDH1A1TSHRMEN1
SCHEMBL23640213 0.56 MEN1 (0.58) MAPK1SMN1; SMN2ESR1ESR2KDM4E
SCHEMBL14604954 0.56 MAOB (0.65) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1996550-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES Novartis AG (CH) 2008-12-03 EP claimed
WO-2007038459-A2 CARBOXYAMINE COMPOUNDS AND THEIR USE IN THE TREATMENT OF HDAC DEPENDENT DISEASES NOVARTIS AG (CH) 2007-04-05 WO claimed