SCHEMBL4777463

SCHEMBL4777463

CC(C)C(=O)Nc1nc(O)c2[nH]cnc2n1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.42
ADORA1 P30542 2/20 0.40
NOS1 P29475 1/20 0.40
NEK2 P51955 4/20 0.39
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HSD17B10 Q99714 1/20 0.38
KDR P35968 2/20 0.38
AURKB Q96GD4 1/20 0.38
CYP1A2 P05177 1/20 0.37
STAT3 P40763 4/20 0.37
ADORA2A P29274 1/20 0.36
CDK1 P06493 2/20 0.35
CCNB1 P14635 2/20 0.35
CCNA2 P20248 2/20 0.35
CDK2 P24941 2/20 0.35
CCNA1 P78396 2/20 0.35
CCNB2 O95067 1/20 0.35
CCNB3 Q8WWL7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9412617 0.86 GDA (0.39) GDANEK2KDRAURKBSTAT3
SCHEMBL4307867 0.84 DPP4 (0.49) GDAADORA1NOS1NEK2ALDH1A1
SCHEMBL887125 0.84 GDA (0.55) GDANEK2KDRAURKBCYP1A2
SCHEMBL30590049 0.78 ADORA1 (0.41) ADORA1NOS1ALDH1A1LMNAHSD17B10
SCHEMBL4777464 0.78 ADORA1 (0.41) ADORA1NOS1ALDH1A1LMNAHSD17B10
SCHEMBL9412640 0.77 GDA (0.39) GDANEK2ALDH1A1KDRAURKB
SCHEMBL377763 0.77 CDK2 (0.48) GDANEK2CDK1CCNB1CCNA2
SCHEMBL19728689 0.75 CDK2 (0.48) ADORA1NOS1ALDH1A1LMNAHSD17B10
SCHEMBL16146261 0.75 ESR1 (0.42) CYP1A2CDK1CCNB1CCNA2CDK2
SCHEMBL12841391 0.74 STAT3 (0.47) NEK2STAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7314923-B2 Nucleoside and oligonucleotide analogues DAIICHI SANKYO COMPANY, LIMITED (JP) 2008-01-01 US claimed
EP-1877057-A1 USE OF PYRAZOLYL-PYRIMIDINE DERIVATIVES IN THE TREATMENT OF PAIN AstraZeneca AB (SE) 2008-01-16 EP disclosed
WO-2006115452-A1 USE OF PYRAZOLYL-PYRIMIDINE DERIVATIVES IN THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2006-11-02 WO disclosed
US-4801710-A Regioselective synthesis of 9-substituted purine acyclonucleoside derivatives MERCK & CO., INC. (US) 1989-01-31 US disclosed
EP-0184473-A1 Regioselective synthesis of 9-substituted purine acyclonucleoside derivatives MERCK & CO. INC. (US) 1986-06-11 EP disclosed