SCHEMBL4777532

SCHEMBL4777532

C[S+]([O-])N(Cc1cccc(Cl)c1Cl)c1ccc(C(C(N)=O)C2CCCNC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 18/20 0.44
SLC6A2 P23975 17/20 0.44
SLC6A3 Q01959 14/20 0.44
KCNH2 Q12809 5/20 0.44
CYP2D6 P10635 5/20 0.44
CYP3A4 P08684 2/20 0.44
OPRK1 P41145 1/20 0.35
REN P00797 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4776759 0.84 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL4777308 0.73 SLC6A4 (0.45) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL5571822 0.71 ALDH1A1 (0.42) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL16475935 0.69 CPN1 (0.47) SLC6A4SLC6A2SLC6A3
SCHEMBL4774929 0.68 SLC6A4 (0.42) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL4792287 0.67 REN (0.38) SLC6A4SLC6A2REN
SCHEMBL4775167 0.65 KDM4E (0.39) KCNH2
SCHEMBL4776560 0.64 RECQL (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6
SCHEMBL27746280 0.62 SLC6A2 (0.48) SLC6A4SLC6A2SLC6A3CYP2D6
SCHEMBL4768070 0.62 SLC6A4 (0.44) SLC6A4SLC6A2SLC6A3KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1942888-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS Cytokinetics, Inc. (US) 2008-07-16 EP disclosed
WO-2007056078-A2 CERTAIN CHEMICAL ENTITIES, COMPOSITIONS, AND METHODS CYTOKINETICS, INC. (US) 2007-05-18 WO disclosed