SCHEMBL4777601

SCHEMBL4777601

N=C(NO)c1cccc2c1Oc1ccccc1C2

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
HDAC4 P56524 2/20 0.34
HDAC7 Q8WUI4 2/20 0.34
HDAC5 Q9UQL6 2/20 0.34
GAA P10253 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC10 Q969S8 1/20 0.31
HDAC11 Q96DB2 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
HDAC9 Q9UKV0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668365 0.81 MAOA (0.50) MAOAMAOBGAANPSR1
SCHEMBL7325719 0.76 MAOA (0.52) MAOAMAOBGAAHDAC8
SCHEMBL4668382 0.75 PARP1 (0.53) MAOAMAOB
SCHEMBL27714413 0.75 TRPA1 (0.54) MAOAMAOBGAANPSR1
SCHEMBL8961832 0.74 MAOA (0.48) MAOAMAOB
SCHEMBL31069904 0.74 MAOA (0.48) MAOAMAOB
SCHEMBL4777607 0.73 MAOA (0.47) MAOAMAOBGAA
SCHEMBL13777196 0.72 MAOA (0.73) MAOAMAOBGAANPSR1
SCHEMBL5094900 0.72 MAOA (0.59) MAOAMAOBGAANPSR1
SCHEMBL11813909 0.72 MAOA (0.59) MAOAMAOBHDAC4HDAC7HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1896467-A2 TRICYCLIC OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V. (BE) 2008-03-12 EP disclosed
WO-2006138528-A2 TRICYCLIC OPIOID MODULATORS JANSSEN PHARMACEUTICA N.V (BE) 2006-12-28 WO disclosed