SCHEMBL4777878

SCHEMBL4777878

CN(C)CCN(C)Cc1c[nH]c2ccc([N+](=O)[O-])cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.53
PKM P14618 1/20 0.47
PKLR P30613 1/20 0.47
SLC6A4 P31645 4/20 0.46
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
HTR1A P08908 3/20 0.44
HTR2A P28223 2/20 0.44
HTR2C P28335 2/20 0.44
MPO P05164 1/20 0.44
HTR7 P34969 2/20 0.44
HTR5A P47898 2/20 0.44
HTR6 P50406 2/20 0.44
POLB P06746 1/20 0.43
HTR1D P28221 4/20 0.43
HTR1B P28222 3/20 0.43
TUBB4A P04350 1/20 0.43
TUBB P07437 1/20 0.43
TUBA3C P0DPH7 1/20 0.43
TUBA1B P68363 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8538163 0.88 NQO2 (0.58) NQO2PKMPKLRSLC6A4MEN1
SCHEMBL2535250 0.86 NQO2 (0.62) NQO2PKMPKLRSLC6A4KMT2A
SCHEMBL7367937 0.85 NQO2 (0.61) NQO2PKMPKLRSLC6A4KMT2A
SCHEMBL3294986 0.80 NQO2 (0.64) NQO2PKMPKLRSLC6A4MEN1
SCHEMBL27929617 0.78 NQO2 (0.61) NQO2PKMPKLRMEN1KMT2A
SCHEMBL4778984 0.78 SLC6A4 (0.68) SLC6A4HTR1AHTR2AHTR2CMPO
SCHEMBL29507879 0.78 PKM (0.63) NQO2PKMPKLRSLC6A4MEN1
SCHEMBL396020 0.78 PKM (0.63) NQO2PKMPKLRSLC6A4MEN1
SCHEMBL11537110 0.76 NQO2 (0.63) NQO2PKMPKLRMEN1KMT2A
SCHEMBL14574202 0.76 GABRP (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1581492-B1 N-ARYLSULFONYL-3-SUBSTITUTED INDOLES HAVING SEROTONIN RECEPTOR AFFINITY, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITION CONTAINING THEM SUVEN LIFE SCIENCES LTD (IN) 2008-07-16 EP disclosed