SCHEMBL4778176

SCHEMBL4778176

NC1C2CN(c3ncccc3Br)CC12

nearest known ligand 0.53

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 2/20 0.34
PTPN11 Q06124 2/20 0.33
TRPV1 Q8NER1 2/20 0.33
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4635199 0.80 HSD11B1 (0.46) MALT1PTPN11TRPV1HSD11B1
SCHEMBL4880417 0.79 PDE10A (0.39) MALT1TRPV1
SCHEMBL4320157 0.76 EPHX2 (0.56) TRPV1HSD11B1
SCHEMBL4635503 0.76 KDM4E (0.54) HSD11B1
SCHEMBL4880388 0.75 ALDH1A1 (0.44) MALT1
SCHEMBL4880724 0.74 KDM4E (0.44) MALT1TRPV1
SCHEMBL4635540 0.74 CYP1A2 (0.62) HSD11B1
SCHEMBL27703385 0.73 CYP1A2 (0.49) MALT1TRPV1
SCHEMBL20406252 0.73 CYP1A2 (0.53) TRPV1
SCHEMBL16496334 0.72 DPP4 (0.43) PTPN11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008010061-A2 3-AZABICYCLO [3.1.0] HEXANE VANILLOID RECEPTOR LIGANDS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM, AND PROCESSES FOR THEIR PREPARATION GLENMARK PHARMACEUTICALS S.A. (US) 2008-01-24 WO disclosed