SCHEMBL4778609

SCHEMBL4778609

N#Cc1c(-c2ccc(N)cc2)[nH]c2cc(O)cc(C3CC3)c12

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 2/20 0.33
ADORA2A P29274 1/20 0.32
ADORA1 P30542 1/20 0.32
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4777353 0.83 MAOA (0.37) IKBKBADORA2AADORA1KDM4EMEN1
SCHEMBL4771469 0.78 TLR9 (0.33) MEN1MAPTKMT2A
SCHEMBL4775583 0.76 PDE10A (0.35) IKBKBKDM4EMEN1ALDH1A1MAPT
SCHEMBL4779519 0.66 TLR9 (0.32)
SCHEMBL27438188 0.61 ALOX5 (0.47) KDM4EMEN1ALDH1A1MAPTHPGD
SCHEMBL15769819 0.60 KDM4E (0.46) IKBKBKDM4EMEN1ALDH1A1MAPT
SCHEMBL10097345 0.60 MAOA (0.50) ADORA1KDM4EMEN1ALDH1A1MAPT
SCHEMBL28819042 0.59 ESR2 (0.60) ADORA2AADORA1KDM4EMEN1ALDH1A1
SCHEMBL1360896 0.59 KDM4E (0.47) KDM4EMEN1ALDH1A1MAPTHPGD
Benzidine SCHEMBL29155805 0.56 CYP3A4 (0.65) MEN1ALDH1A1MAPTKMT2AHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1984332-A2 METHODS FOR TREATING HEPATITIS C PTC Therapeutics, Inc. (US) 2008-10-29 EP disclosed
WO-2007084413-A2 METHODS FOR TREATING HEPATITIS C PTC THERAPEUTICS, INC. (US) 2007-07-26 WO disclosed