SCHEMBL4779658

SCHEMBL4779658

COc1ccc(CC=O)c(C)c1C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
ALDH1A1 P00352 4/20 0.47
TSHR P16473 3/20 0.47
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
NR3C1 P04150 1/20 0.38
PGR P06401 1/20 0.38
NR3C2 P08235 1/20 0.38
IMPDH2 P12268 1/20 0.38
POLB P06746 1/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
HSD17B10 Q99714 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
BMP1 P13497 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5610695 0.89 MEN1 (0.44) MEN1KMT2AALDH1A1TSHRLMNA
SCHEMBL5495434 0.84 ALDH1A1 (0.38) MEN1KMT2AALDH1A1TSHRNR3C1
SCHEMBL578043 0.84 ALDH1A1 (0.41) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL4781858 0.81 FDPS (0.38) MEN1KMT2AALDH1A1TSHRMAPT
SCHEMBL7151009 0.81 AOC3 (0.49) MEN1KMT2AALDH1A1TSHRLMNA
SCHEMBL5241041 0.80 ALDH1A1 (0.44) MEN1KMT2AALDH1A1TSHRLMNA
SCHEMBL2730801 0.80 ALDH1A1 (0.41) MEN1KMT2AALDH1A1LMNAMAPT
SCHEMBL5290521 0.79 MEN1 (0.53) MEN1KMT2AALDH1A1TSHRLMNA
Formaldehyde SCHEMBL5244081 0.78 ALDH1A1 (0.42) MEN1KMT2AALDH1A1TSHRLMNA
SCHEMBL24541830 0.77 CA1 (0.40) MEN1KMT2AALDH1A1TSHRPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008016811-A2 AMINOPIPERIDINES AND REALTED COMPOUNDS NEUROGEN CORPORATION (US) 2008-02-07 WO disclosed
EP-1756107-A2 ARYL-SUBSTITUTED PIPERAZINE DERIVATIVES NEUROGEN CORPORATION (US) 2007-02-28 EP disclosed
WO-2006009789-A2 ARYL-SUBSTITUTED PIPERAZINE DERIVATIVES NEUROGEN CORPORATION (US) 2006-01-26 WO disclosed
WO-2005110982-A2 SUBSTITUTED 1-BENZYL-4-SUBSTITUTED PIPERAZINE ANALOGUES NEUROGEN CORPORATION (US) 2005-11-24 WO disclosed