SCHEMBL5495434

SCHEMBL5495434

COc1ccc(CC=O)c(F)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.38
MEN1 O00255 4/20 0.37
KMT2A Q03164 4/20 0.37
TSHR P16473 3/20 0.37
TAAR1 Q96RJ0 1/20 0.37
TUBB1 Q9H4B7 2/20 0.35
HPGD P15428 3/20 0.35
POLB P06746 1/20 0.35
HSD17B10 Q99714 2/20 0.34
KDM4E B2RXH2 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
CYP1A2 P05177 1/20 0.34
GLA P06280 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
PKM P14618 1/20 0.34
CYP2C19 P33261 1/20 0.34
RECQL P46063 1/20 0.34
NR3C1 P04150 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4779658 0.84 MEN1 (0.47) ALDH1A1MEN1KMT2ATSHRTAAR1
SCHEMBL5165930 0.83 ALDH1A1 (0.40) ALDH1A1MEN1KMT2ATSHRTAAR1
SCHEMBL5610695 0.81 MEN1 (0.44) ALDH1A1MEN1KMT2ATSHRTAAR1
SCHEMBL578043 0.79 ALDH1A1 (0.41) ALDH1A1MEN1KMT2ATSHRHPGD
SCHEMBL25388605 0.79 ALDH1A1 (0.38) ALDH1A1MEN1KMT2ATSHRTUBB1
SCHEMBL13859482 0.79 TDP1 (0.46) ALDH1A1MEN1KMT2AHPGDPOLB
SCHEMBL577619 0.78 ALDH1A1 (0.37) ALDH1A1MEN1KMT2ATSHRTUBB1
SCHEMBL16794991 0.77 HTR2A (0.45) ALDH1A1KMT2ATAAR1L3MBTL1
SCHEMBL2689127 0.75 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ATSHRHPGD
SCHEMBL30536248 0.75 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ATSHRHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765760-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F.HOFFMANN-LA ROCHE AG (CH) 2007-03-28 EP disclosed
WO-2006002802-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO disclosed