SCHEMBL4779942

SCHEMBL4779942

COc1cc2nc(-c3cccc(NCc4cccnc4)c3)nc(Nc3ccc4c(cnn4C(=O)OC(C)(C)C)c3)c2cc1O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.44
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 2/20 0.44
EEF2K O00418 1/20 0.44
MAP4K4 O95819 1/20 0.44
CLK2 P49760 1/20 0.44
GSK3B P49841 1/20 0.44
PRKX P51817 1/20 0.44
NEK4 P51957 1/20 0.44
PRKG2 Q13237 1/20 0.44
PKN2 Q16513 1/20 0.44
TAOK1 Q7L7X3 1/20 0.44
AURKB Q96GD4 1/20 0.44
PBK Q96KB5 1/20 0.44
SLK Q9H2G2 1/20 0.44
MAP3K20 Q9NYL2 1/20 0.44
EGFR P00533 3/20 0.43
ITK Q08881 1/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780062 0.92 EGFR (0.42) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL1729245 0.91 MEN1 (0.45) CLK4ROCK2EGFRMEN1KMT2A
SCHEMBL4784662 0.91 EGFR (0.43) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL4798787 0.90 ROCK2 (0.46) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL3793329 0.89 ABCG2 (0.54) ROCK2EGFRITKTSHRABCG2
SCHEMBL877065 0.87 EGFR (0.45) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL4783152 0.86 EGFR (0.43) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL877114 0.86 ABCG2 (0.45) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL877064 0.86 ROCK2 (0.51) CLK4ROCK2ROCK1EEF2KMAP4K4
SCHEMBL877115 0.84 ABCG2 (0.47) CLK4ROCK2ROCK1EEF2KMAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008054599-A2 RHO KINASE INHIBITORS SURFACE LOGIX, INC. (US) 2008-05-08 WO disclosed
EP-1865958-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS Surface Logix, Inc. (US) 2007-12-19 EP disclosed
WO-2006105081-A2 PHARMACOKINETICALLY IMPROVED COMPOUNDS SURFACE LOGIX, INC. (US) 2006-10-05 WO disclosed