SCHEMBL4779949

SCHEMBL4779949

COc1c(C#N)cc(C(C)(C)C)cc1NC(=O)c1cnc(C)c(-n2cc(C(=O)NN3CCCCC3)nn2)c1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 6/20 0.37
BRAF P15056 7/20 0.35
THRB P10828 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CNR1 P21554 1/20 0.31
RORC P51449 1/20 0.31
NR1I2 O75469 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781871 0.90 MAPK14 (0.37) MAPK14BRAFCNR1
SCHEMBL4902142 0.87 BRAF (0.48) MAPK14BRAF
SCHEMBL4782271 0.86 MAPK14 (0.39) MAPK14BRAFNR1I2
SCHEMBL4781875 0.86 SCN10A (0.34) MAPK14BRAFKDM4EALDH1A1CNR1
SCHEMBL4782863 0.84 NR1I2 (0.40) MAPK14BRAFCNR1NR1I2
SCHEMBL4783254 0.78 MAPK14 (0.35) MAPK14
SCHEMBL4780817 0.77 NR1I2 (0.36) CNR1NR1I2
SCHEMBL4467266 0.77 MAPK14 (0.41) MAPK14BRAF
SCHEMBL1378709 0.75 MAPK14 (0.39) MAPK14BRAF
SCHEMBL4783260 0.74 MAPK14 (0.31) MAPK14BRAFNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed