SCHEMBL4779984

SCHEMBL4779984

Cc1ncc(Nc2cc(F)cc(N3CCOCC3)c2)cc1-n1cc(C(=O)NCC2CCCO2)nn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.41
GLS O94925 2/20 0.39
PLAU P00749 1/20 0.39
POLB P06746 2/20 0.38
TNK2 Q07912 1/20 0.38
ATM Q13315 2/20 0.38
TSHR P16473 1/20 0.37
ALDH1A1 P00352 3/20 0.37
HPGD P15428 3/20 0.37
RAB9A P51151 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
TP53 P04637 2/20 0.37
NPC1 O15118 1/20 0.37
BRAF P15056 2/20 0.37
MAPT P10636 1/20 0.37
PDE10A Q9Y233 1/20 0.36
KDM4E B2RXH2 1/20 0.36
CYP1A2 P05177 1/20 0.36
GAA P10253 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781496 0.98 ACKR3 (0.40) ACKR3GLSPLAUPOLBTNK2
SCHEMBL4783075 0.91 PLAU (0.42) ACKR3PLAUBRAF
SCHEMBL4778219 0.90 NAPEPLD (0.40) ACKR3PLAUBRAFCYP1A2CYP2C19
SCHEMBL4782767 0.90 CNR2 (0.42) ACKR3GLSPLAUBRAFCYP1A2
SCHEMBL4783684 0.90 ACKR3 (0.40) ACKR3GLSPOLBATMALDH1A1
SCHEMBL4781500 0.89 PLAU (0.41) ACKR3PLAUBRAF
SCHEMBL4936382 0.86 HPGD (0.41) ACKR3GLSPOLBATMALDH1A1
SCHEMBL4780823 0.86 ACKR3 (0.39) ACKR3GLSTNK2ATMALDH1A1
SCHEMBL4781359 0.84 ACKR3 (0.47) ACKR3PLAUBRAFGAA
SCHEMBL4780831 0.84 TNK2 (0.39) ACKR3GLSTNK2ALDH1A1BRAF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed