SCHEMBL4782767

SCHEMBL4782767

Cc1ncc(Nc2cc(F)cc(N3CCOCC3)c2)cc1-n1cc(C(=O)NCC2CCOCC2)nn1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 5/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.42
PLAU P00749 1/20 0.39
NAPEPLD Q6IQ20 1/20 0.38
ACKR3 P25106 2/20 0.38
GLS O94925 3/20 0.37
AOC2 O75106 1/20 0.37
PIK3CB P42338 1/20 0.36
BRAF P15056 5/20 0.36
RAF1 P04049 3/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
MAPK14 Q16539 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4778219 0.98 NAPEPLD (0.40) CNR2CYP2D6CYP2C19CYP1A2PLAU
SCHEMBL4779984 0.90 ACKR3 (0.41) CYP2C19CYP1A2PLAUACKR3GLS
SCHEMBL4778221 0.88 RAF1 (0.43) PLAUBRAFRAF1MAPK14
SCHEMBL4781496 0.88 ACKR3 (0.40) PLAUACKR3GLSBRAF
SCHEMBL4782171 0.86 PLAU (0.38) PLAUBRAFRAF1MAPK14
SCHEMBL4780442 0.86 PLAU (0.38) PLAUBRAFRAF1
SCHEMBL4781149 0.85 PLAU (0.40) PLAUBRAFRAF1MAPK14
SCHEMBL4781359 0.85 ACKR3 (0.47) CNR2PLAUACKR3BRAFRAF1
SCHEMBL4782308 0.85 PLAU (0.41) PLAUBRAFRAF1MAPK14
SCHEMBL4783670 0.83 MAPK14 (0.39) PLAUPIK3CBBRAFRAF1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed