SCHEMBL4781607

SCHEMBL4781607

Cc1ncc(Nc2cc(C#N)cc(C(C)(C)C)c2)cc1-n1cc(C(=O)NC2CCCCC2)nn1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 6/20 0.41
NR1I2 O75469 1/20 0.36
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
PRKAA2 P54646 2/20 0.34
GPR119 Q8TDV5 1/20 0.34
CNR2 P34972 2/20 0.34
CNR1 P21554 1/20 0.34
PDE7A Q13946 2/20 0.33
GLS O94925 1/20 0.33
TSHR P16473 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
TYK2 P29597 1/20 0.33
STAT3 P40763 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4780707 0.93 NR1I2 (0.36) ACKR3NR1I2PRKAA2GPR119IRAK4
SCHEMBL4779570 0.92 SSTR4 (0.40) ACKR3NR1I2PRKAA2GPR119
SCHEMBL4781611 0.90 TEK (0.39) ACKR3NR1I2NPC1RAB9APRKAA2
SCHEMBL4780817 0.86 NR1I2 (0.36) NR1I2GPR119CNR2CNR1IRAK4
SCHEMBL4782033 0.86 NR1I2 (0.35) NR1I2GPR119IRAK4TYK2STAT3
SCHEMBL4782188 0.84 MEN1 (0.42) ACKR3NR1I2
SCHEMBL4779207 0.84 NR1I2 (0.38) ACKR3NR1I2GPR119CNR2IRAK4
SCHEMBL4780719 0.83 TEK (0.39) ACKR3NR1I2PRKAA2GPR119
SCHEMBL4781558 0.83 GLS (0.41) ACKR3NPC1RAB9AGLSSMN1; SMN2
SCHEMBL4783140 0.82 MAPK14 (0.36) NR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed