SCHEMBL4779207

SCHEMBL4779207

Cc1ncc(Nc2cc(C#N)cc(C(C)(C)C)c2)cc1-n1cc(C(=O)NCC(C)(C)C)nn1

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.38
KLKB1 P03952 1/20 0.33
USP30 Q70CQ3 1/20 0.33
TEK Q02763 2/20 0.32
GPR119 Q8TDV5 2/20 0.32
CNR2 P34972 1/20 0.32
DDT P30046 3/20 0.31
IRAK4 Q9NWZ3 2/20 0.31
MIF P14174 1/20 0.31
ACKR3 P25106 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4783774 0.93 NR1I2 (0.36) NR1I2KLKB1USP30TEKGPR119
SCHEMBL4782660 0.90 NR1I2 (0.42) NR1I2KLKB1USP30TEKDDT
SCHEMBL4783414 0.90 NR1I2 (0.35) NR1I2USP30GPR119CNR2IRAK4
SCHEMBL4780027 0.89 NR1I2 (0.36) NR1I2KLKB1USP30TEKGPR119
SCHEMBL4779210 0.89 TEK (0.41) NR1I2TEKDDTMIF
SCHEMBL4782188 0.86 MEN1 (0.42) NR1I2ACKR3
SCHEMBL4778554 0.86 DDT (0.42) NR1I2DDT
SCHEMBL4782621 0.86 GLS (0.43) NR1I2KLKB1MIF
SCHEMBL4782886 0.85 NR1I2 (0.38) NR1I2GPR119IRAK4
SCHEMBL4782867 0.85 NR1I2 (0.36) NR1I2KLKB1USP30GPR119DDT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed