Pyrene

Pyrene

SCHEMBL4782088

C[C@H](N)C(=O)O.c1cc2ccc3cccc4ccc(c1)c2c34

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.50
MEN1 O00255 3/20 0.50
ALDH1A1 P00352 6/20 0.48
HSD17B10 Q99714 5/20 0.48
HPGD P15428 4/20 0.48
TSHR P16473 3/20 0.48
CYP1A2 P05177 2/20 0.48
CYP3A4 P08684 2/20 0.48
CYP1A1 P04798 1/20 0.48
CYP1B1 Q16678 1/20 0.48
KDM4E B2RXH2 7/20 0.44
GAA P10253 1/20 0.44
CASP1 P29466 1/20 0.44
CASP7 P55210 1/20 0.44
MAPT P10636 1/20 0.42
GLA P06280 1/20 0.40
POLB P06746 1/20 0.40
CYP2D6 P10635 1/20 0.40
XIAP P98170 1/20 0.40
BIRC2 Q13490 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naphthalene SCHEMBL699807 0.84 TAAR1 (0.46) ALDH1A1CYP1A2KDM4ECYP2D6XIAP
Naphthalene SCHEMBL699808 0.84 TAAR1 (0.46) ALDH1A1CYP1A2KDM4ECYP2D6XIAP
Alanine SCHEMBL28922813 0.79 ELANE (0.42) ALDH1A1CYP1A2KDM4EMAPTXIAP
Pyrene SCHEMBL6033008 0.79 ALDH1A1 (0.61) KMT2AMEN1ALDH1A1HSD17B10HPGD
Anthracene SCHEMBL29064584 0.78 EPHX1 (0.44) KMT2AMEN1ALDH1A1HSD17B10HPGD
Pyrene SCHEMBL21599111 0.78 ALDH1A1 (0.69) KMT2AMEN1ALDH1A1HSD17B10HPGD
Alanine SCHEMBL21616532 0.78 SLC7A5 (0.53) ALDH1A1MAPTXIAPTAAR1
Alanine SCHEMBL27615995 0.78 SLC7A5 (0.53) ALDH1A1MAPTXIAPTAAR1
Pyrene SCHEMBL27931631 0.77 ALDH1A1 (0.58) KMT2AMEN1ALDH1A1HSD17B10HPGD
SCHEMBL5593608 0.76 AKR1B1 (0.60) KMT2AMEN1ALDH1A1HSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008003773-A1 METHOD FOR DETECTING INTERACTIONS USING THE FLUORESCENCE REPORTER PYRENYLALANINE PHARMALEADS (FR) 2008-01-10 WO disclosed