SCHEMBL4782298

SCHEMBL4782298

CC(=O)Cn1cc(C(=O)NCC(C)(C)C)nn1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 1/20 0.40
GLS O94925 6/20 0.39
KLKB1 P03952 3/20 0.37
CYP2C19 P33261 1/20 0.36
GLA P06280 1/20 0.36
MAPK1 P28482 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35
CNR2 P34972 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4781660 0.81 GLS (0.41) GLS
SCHEMBL22247229 0.76 GLA (0.40) SMYD3GLAMAPK1ALDH1A1LMNA
SCHEMBL21206316 0.71 SMYD3 (0.40) SMYD3GLSCYP2C19GLAMAPK1
SCHEMBL24125043 0.70 SMYD3 (0.37) SMYD3GLSCYP2C19GLAMAPK1
SCHEMBL8931483 0.70 HRH4 (0.41) GLAALDH1A1LMNA
SCHEMBL24621692 0.68 TSHR (0.40) SMYD3GLAMAPK1ALDH1A1LMNA
SCHEMBL25447017 0.68 GLS (0.38) SMYD3GLSCYP2C19GLAMAPK1
SCHEMBL11910527 0.68 SRC (0.41) GLAMAPK1ALDH1A1LMNACNR2
SCHEMBL31720484 0.68 SMYD3 (0.41) SMYD3GLSKLKB1GLAMAPK1
SCHEMBL7963203 0.67 NOTUM (0.49) GLS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed
WO-2008021388-A1 HETEROARYL DERIVATIVES AS CYTOKINE INHIBITORS KEMIA, INC. (US) 2008-02-21 WO disclosed