SCHEMBL4783216

SCHEMBL4783216

OCC1c2ccccc2CCN1c1nc(-c2cccc(O)c2)nc(N2CCN(C3CCCCC3)CC2)n1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 7/20 0.45
ESR2 Q92731 5/20 0.45
PIK3CA P42336 6/20 0.39
KDM2B Q8NHM5 1/20 0.39
ESRRG P62508 3/20 0.37
ESRRA P11474 2/20 0.37
MTOR P42345 1/20 0.37
ESRRB O95718 1/20 0.36
SIGMAR1 Q99720 4/20 0.36
HPGD P15428 1/20 0.35
HSD17B10 Q99714 1/20 0.35
PIK3CD O00329 1/20 0.35
PIK3CB P42338 1/20 0.35
PIK3CG P48736 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4785905 0.99 ESR1 (0.44) ESR1ESR2PIK3CAKDM2BESRRG
SCHEMBL4786261 0.91 PIK3CA (0.46) ESR1ESR2PIK3CAMTORPIK3CG
SCHEMBL4783015 0.88 PIK3CA (0.48) PIK3CAMTORPIK3CG
SCHEMBL4782297 0.87 PIK3CA (0.43) ESR1ESR2PIK3CAMTOR
SCHEMBL4783923 0.87 HRH4 (0.43) ESR1ESR2PIK3CAMTOR
SCHEMBL4884094 0.86 PIK3CA (0.44) ESR1ESR2PIK3CAMTORPIK3CB
SCHEMBL4784160 0.86 PIK3CA (0.42) ESR1ESR2PIK3CAMTOR
SCHEMBL4784640 0.86 ADORA3 (0.43) ESR1ESR2PIK3CAMTORPIK3CG
SCHEMBL4784132 0.85 PIK3CA (0.44) ESR1ESR2PIK3CAMTOR
SCHEMBL4784088 0.85 PIK3CA (0.43) ESR1ESR2PIK3CAMTORHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed