SCHEMBL4783447

SCHEMBL4783447

NC(=O)C1CCN(Cc2ccc3ccc(=O)oc3c2)CC1

nearest known ligand 0.64

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 13/20 0.64
DRD2 P14416 8/20 0.64
KCNH2 Q12809 1/20 0.56
MCHR2 Q969V1 1/20 0.56
MCHR1 Q99705 1/20 0.56
CYP19A1 P11511 1/20 0.50
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8431212 0.78 DRD4 (1.00) DRD4DRD2
SCHEMBL8435196 0.77 DRD4 (1.00) DRD4DRD2CYP19A1
SCHEMBL8432504 0.76 DRD4 (0.79) DRD4DRD2KCNH2MCHR2MCHR1
SCHEMBL6333889 0.73 MCHR1 (1.00) KCNH2MCHR2MCHR1
SCHEMBL16582078 0.73 ALDH1A1 (0.64) KCNH2KDM4EALDH1A1
SCHEMBL5368002 0.73 GAA (0.69) DRD4DRD2KDM4EALDH1A1
SCHEMBL12660139 0.73 KDM4E (0.64) KCNH2KDM4EALDH1A1
SCHEMBL8431223 0.72 DRD4 (1.00) DRD4DRD2KDM4EALDH1A1
SCHEMBL26133908 0.72 ICAM1 (0.52) KCNH2KDM4EALDH1A1
SCHEMBL14174789 0.72 ALDH1A1 (0.67) KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008045564-A2 CARBOXAMIDE COMPOUNDS AND THEIR USE AS ANTAGONISTS OF THE CHEMOKINE CCR2 RECEPTOR EPIX DELAWARE, INC. (US) 2008-04-17 WO claimed