SCHEMBL4783608

SCHEMBL4783608

CC(C)(C)OC(=O)NCCCn1cccc1C(=O)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.49
MEN1 O00255 2/20 0.48
MAPT P10636 2/20 0.48
KMT2A Q03164 2/20 0.48
LMNA P02545 1/20 0.48
ALOX12 P18054 1/20 0.48
RECQL P46063 1/20 0.48
DRD2 P14416 4/20 0.47
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
SIGMAR1 Q99720 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
GAA P10253 1/20 0.43
TP53 P04637 1/20 0.43
BRD4 O60885 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27246689 0.83 TDP1 (0.52) MEN1KMT2ADRD2SIGMAR1TDP1
SCHEMBL3953782 0.83 NPC1 (0.40) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL3387585 0.77 DRD2 (0.47) MEN1KMT2ADRD2SIGMAR1TDP1
SCHEMBL6675697 0.76 DRD2 (0.46) MEN1KMT2ADRD2SIGMAR1TDP1
SCHEMBL20386735 0.75 DRD2 (0.48) MAPTDRD2SIGMAR1
SCHEMBL1308684 0.75 DRD2 (0.55) DRD2SIGMAR1TDP1
SCHEMBL10374343 0.74 PPARG (0.41) ALDH1A1MEN1MAPTKMT2ALMNA
SCHEMBL3388119 0.74 DRD2 (0.44) MEN1MAPTKMT2ALMNADRD2
SCHEMBL1467340 0.74 NAAA (0.56) ALDH1A1MEN1KMT2ALMNANPC1
SCHEMBL4782988 0.74 CNR2 (0.47) DRD2SIGMAR1TDP1BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008067222-A1 HETEROCYCLIC MODULATORS OF TGR5 KALYPSYS, INC. (US) 2008-06-05 WO disclosed