SCHEMBL4784475

SCHEMBL4784475

CCOc1cc(-c2cccc(N)n2)ccc1OCC[As](C)C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.45
PDE4A P27815 1/20 0.42
PDE4B Q07343 1/20 0.42
PDE4C Q08493 1/20 0.42
PDE4D Q08499 1/20 0.42
S1PR1 P21453 5/20 0.41
NOS3 P29474 3/20 0.41
NOS1 P29475 3/20 0.41
S1PR3 Q99500 1/20 0.41
CTSS P25774 1/20 0.40
FPR2 P25090 1/20 0.40
KDM4E B2RXH2 4/20 0.40
HSD17B10 Q99714 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
NOS2 P35228 1/20 0.40
MAPT P10636 3/20 0.38
MEN1 O00255 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL220774 0.83 NOS1 (0.60) MAOBS1PR1NOS3NOS1S1PR3
SCHEMBL221746 0.80 NOS3 (0.60) S1PR1NOS3NOS1S1PR3ALDH1A1
SCHEMBL221745 0.76 FPR2 (0.39) MAOBS1PR1NOS3NOS1FPR2
SCHEMBL221219 0.72 NOS1 (0.71) NOS3NOS1KDM4EALDH1A1NPC1
SCHEMBL220877 0.69 NOS3 (0.61) NOS3NOS1NOS2
SCHEMBL221744 0.69 FPR2 (0.38) MAOBPDE4DS1PR1NOS3NOS1
SCHEMBL219485 0.68 NOS3 (0.64) NOS3NOS1CTSSNOS2
SCHEMBL8082378 0.68 NOS1 (0.57) NOS3NOS1NOS2
SCHEMBL1965584 0.66 PDE4A (0.65) PDE4APDE4BPDE4CPDE4DS1PR1
SCHEMBL1778039 0.66 HSD17B10 (0.65) S1PR1S1PR3KDM4EHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008073451-A2 BENZOIMIDAZOLE DERIVATIVES AS SIRTUIN (SIR) MODULATING COMPOUNDS SIRTRIS PHARMACEUTICALS, INC. (US) 2008-06-19 WO disclosed