SCHEMBL4785260

SCHEMBL4785260

O=C1CCCCN1c1ccc[nH]c1=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.40
AURKB Q96GD4 1/20 0.40
INCENP Q9NQS7 1/20 0.40
PARP1 P09874 5/20 0.38
HSD17B10 Q99714 2/20 0.37
GFER P55789 1/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
DAO P14920 1/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TP53 P04637 1/20 0.35
MAPT P10636 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
AKR1C3 P42330 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL924443 0.95 HSD17B10 (0.41) AURKAAURKBINCENPPARP1HSD17B10
SCHEMBL28271187 0.78 ALDH1A1 (0.39) AURKAAURKBINCENPPARP1HSD17B10
SCHEMBL21383788 0.78 SMN1; SMN2 (0.45) ALDH1A1HPGDTP53MAPTL3MBTL1
SCHEMBL9234686 0.77 MAPT (0.46) AURKAAURKBINCENPGFERDAO
SCHEMBL1439000 0.76 GFER (0.44) HSD17B10GFERAPOBEC3AAPOBEC3GALDH1A1
SCHEMBL28807259 0.75 MAPT (0.49) AURKAAURKBINCENPGFERDAO
SCHEMBL30088186 0.75 HTR6 (0.39) PARP1HSD17B10GFERAPOBEC3AAPOBEC3G
SCHEMBL21805200 0.75 HTR6 (0.39) PARP1HSD17B10GFERAPOBEC3AAPOBEC3G
SCHEMBL10751956 0.74 ALDH1A1 (0.42) AURKAAURKBINCENPHSD17B10ALDH1A1
SCHEMBL28834312 0.74 KEAP1 (0.53) HSD17B10GFERAPOBEC3AAPOBEC3GALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008074450-A2 NON-PEPTIDIC RENIN INHIBITORS NITRODERIVATIVES NICOX S.A. (FR) 2008-06-26 WO claimed
WO-2008074450-A2 NON-PEPTIDIC RENIN INHIBITORS NITRODERIVATIVES NICOX S.A. (FR) 2008-06-26 WO disclosed