SCHEMBL4785269

SCHEMBL4785269

CN1C2CCC1CC(OC(=O)c1cccn1C)C2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 4/20 0.63
HTR3B O95264 4/20 0.63
HTR3A P46098 4/20 0.63
HTR3D Q70Z44 4/20 0.63
HTR3C Q8WXA8 4/20 0.63
CHRNA7 P36544 2/20 0.63
CYP2D6 P10635 4/20 0.56
CYP2C19 P33261 2/20 0.56
LMNA P02545 2/20 0.56
CYP1A2 P05177 2/20 0.55
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
NR1I2 O75469 1/20 0.55
MTOR P42345 2/20 0.53
CHRM5 P08912 2/20 0.53
CHRM1 P11229 2/20 0.53
CHRM3 P20309 2/20 0.53
GMNN O75496 1/20 0.53
ALOX15 P16050 1/20 0.53
TSHR P16473 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30621986 0.79 MAPT (0.41) TSHRMAPTSLC6A4KCNH2
SCHEMBL7281727 0.79 KCNH2 (0.55) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7652481 0.79 HTR3A (0.75) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7652475 0.79 HTR3A (0.75) HTR3EHTR3BHTR3AHTR3DHTR3C
Benzoyl Tropine SCHEMBL1103723 0.78 HTR3E (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Benzoyl Tropine SCHEMBL30954638 0.78 HTR3E (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Benzoyl Tropine SCHEMBL221830 0.78 HTR3E (1.00) HTR3EHTR3BHTR3AHTR3DHTR3C
Benzoyl Tropine SCHEMBL3498565 0.77 HTR3E (0.97) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL6506216 0.74 HTR3A (0.63) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL5789144 0.74 HTR3A (0.68) HTR3EHTR3BHTR3AHTR3DHTR3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008098329-A2 PHARMACEUTICAL COMPOSITION, PHARMACEUTICAL PRODUCT, OBTAINING PROCESSES OF PHARMACEUTICAL COMPOUNDS AND USE OF SUCH COMPOUNDS FOR TREATING ERECTILE DYSFUNCTION ACHÉ LABORATÓRIOS FARMACÊUTICOS S/A (BR) 2008-08-21 WO disclosed