SCHEMBL4786376

SCHEMBL4786376

O=C(C1CCCO1)N1CCN(c2nc(-c3cccc(O)c3)nc(N3Cc4ccccc4C[C@@H]3CO)n2)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 7/20 0.45
ALDH1A1 P00352 5/20 0.45
HSD17B10 Q99714 4/20 0.45
TSHR P16473 2/20 0.45
NAMPT P43490 4/20 0.44
HPGD P15428 4/20 0.43
GLA P06280 4/20 0.43
GAA P10253 3/20 0.43
MAPK1 P28482 2/20 0.43
HTT P42858 2/20 0.43
TP53 P04637 1/20 0.43
SLC22A1 O15245 1/20 0.43
ABCC4 O15439 1/20 0.43
LMNA P02545 1/20 0.43
ADRA2A P08913 1/20 0.43
ADRA2B P18089 1/20 0.43
ADRA2C P18825 1/20 0.43
DRD1 P21728 1/20 0.43
ACHE P22303 1/20 0.43
ADRA1D P25100 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4848943 0.84 PIK3CA (0.47) ALDH1A1HSD17B10TSHRHPGDMAPK1
SCHEMBL4785892 0.84 PIK3CA (0.47) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL4786374 0.84 KDM4E (0.44) KDM4EALDH1A1HSD17B10TSHRNAMPT
SCHEMBL4782727 0.82 PIK3CA (0.58) KMT2APIK3CA
SCHEMBL4785240 0.82 PIK3CA (0.58) KMT2APIK3CA
SCHEMBL4784749 0.81 PIK3CA (0.42) ALDH1A1GAALMNAPIK3CA
SCHEMBL4785845 0.81 HRH4 (0.44) SMN1; SMN2PIK3CA
SCHEMBL4846093 0.81 HRH4 (0.44) SMN1; SMN2PIK3CA
SCHEMBL4782301 0.81 PIK3CA (0.43) MEN1KMT2APIK3CA
SCHEMBL4783926 0.81 HRH4 (0.44) SMN1; SMN2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO claimed
WO-2008072850-A1 TRIAZINE DERIVATIVES HAVING INHIBITORY ACTIVITY AGAINST ACETYL-COA CARBOXYLASE AMOREPACIFIC CORPORATION (KR) 2008-06-19 WO disclosed